Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9891 |
PARP1-IN-8
N-(3-chlorophenyl)-3-(1-oxo-4-phenylphthalazin-2(1H)-yl)propanamide |
PARP | Chromatin/Epigenetic; DNA Damage/DNA Repair |
PARP1-IN-8 (N-(3-chlorophenyl)-3-(1-oxo-4-phenylphthalazin-2(1H)-yl)propanamide) 是PARP1的有效抑制剂(IC50 = 97 nM)。 | |||
T79364 |
Antiangiogenic agent 4
|
Akt | Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Antiangiogenic agent 4(Compound 3b)在HFF和HUVEC细胞中抑制Akt磷酸化,可应用于癌症研究。 |